Panitch Schwarze Belisario & Nadel LLP
Pyrrole six-membered heteroaryl ring derivative, preparation method thereof, and medicinal uses thereof
The present invention relates to a pyrrole six-membered heteroaryl ring derivative, the preparation method therefor, and the medicinal uses thereof. Specifically, the present invention relates to a new pyrrole six-membered heteroaryl ring derivative as represented by formula (I), the preparation method therefor, a medicinal composition comprising the derivative, and a therapeutic method using same, and, in particular, the uses as a JAK inhibitor and an immunosuppressor. Substituents in formula (I) have the same definitions as in the description.
Shanghai Hengrui Pharmaceutical Co., Ltd. Jiangsu Hengrui Medicine Co., Ltd.
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Xiaotao Yaoping Xuejun Jiong Qing Bonian
Li Zhu Zhang Lan Dong Liu