Scully, Scott, Murphy & Presser, P.C.
EZH2 inhibitor and use thereof
An inhibitor of a wild type and Y641F mutant of human histone methyltransferase EZH2 is provided herein. Particularly, the inhibitor is a compound represented by formula (I) or a pharmaceutically acceptable salt thereof. The inhibitor can be used to treat a cancer or precancerous condition related to EZH2 activity.
TARAPEUTICS SCIENCE INC.
A A C A A A C C C C A A C C A A
A61K A61P C07D A61K A61P A61K C07D C07D C07D C07D A61K A61K C07D C07D A61K A61K
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Fengchao Bei Lei Chen Wen Liang Li Wen Chao Ao Li Zi Ping Xiao Fei Tao Jing Qingsong
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