Birch, Stewart, Kolasch & Birch, LLP
2, 3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredient
The invention refers to novel 2,3-benzodiazepine derivatives of formula (I) and pharmaceutical compositions containing the same as the active ingredient. The novel compounds antipasmodic, muscle relaxant and neuroprotective activities. In formula I; X represents a hydrogen atom, a chloro atom or a methoxy group; Y stands for a hydrogen atom or a halo atom; Z means a methyl group or a chloro atom; R is a C1-4 alkyl group or a group of the formula —NR1R2, wherein R1 and R2 represent, independently, a hydrogen atom, a C1-4 alkyl group, a C1-4 alkoxy group or a C3-6 cycloalkyl group.
Egis Gyogyszergyar RT.
A A A A A A A C A A A A A A
A61P A61P A61P A61P A61P A61P A61P C07D A61P A61P A61P A61P A61P A61P
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Gyula Gábor László  Gábor Bernadett István Zoltán Gábor Zoltán Miklós Géza József György
Simig Gigler Hársing Martonné Markó Ling Rátkai Szénási Greff Végh Szabó Barkóczy Lévay