Fox Rothschild LLP
Tricyclic Gyrase inhibitors
Disclosed herein are compounds having the structure of Formula I and pharmaceutically suitable salts, esters, and prodrugs thereof that are useful as antibacterially effective tricyclic gyrase inhibitors. In addition, species of tricyclic gyrase inhibitors compounds are also disclosed herein.Related pharmaceutical compositions, uses and methods of making the compounds are also contemplated.
LAWRENCE LIVERMORE NATIONAL SECURITY, LLC MERCK SHARP & DOHME CORP.
C C C C A C C
C07D C07D C07D C07D A61P C07D C07D
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Min Allen Daniel Felice C. Leslie William Suk Joong Thanh To Toan B. Xiaoming John M. Zhiyong Junhu Michael E. Michael Sergio E.
Teng Borchardt Bensen Lightstone Tari Lee Lam Nguyen Li Finn Chen Zhang Jung Trzoss Wong