Cooley LLP
Salt form of a human histone methyltransferase EZH2 inhibitor
Provided herein is N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl (tetrahydro-2H-pyran-4-yl)amino)-4-methyl-4′-(morpholinomethyl)-[1,1′-biphenyl]-3-carboxamide hydrobromide. Also provided herein is a particular polymorph form of this compound.
Epizyme, Inc. Eisai R&D Management Co., Ltd.
Y A A C C
Y02A A61P A61K C07D C07D
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Steven Arani Kristen Hyeong Wook Kuan-Chun Frances Kevin Wayne
Mathieu Chanda Sanders Choi Huang Fang Kuntz