McCarter & English, LLP
Galunisertib crystalline form, preparation method thereof and use thereof
The present disclosure relates to a novel crystalline form of Galunisertib, processes for preparation and use thereof. The present disclosure also relates to a pharmaceutical composition comprises the novel crystalline form of Galunisertib and use of the novel crystalline form of Galunisertib and pharmaceutical composition for preparing drugs treating disease. The crystalline form of the present disclosure has good stability, solubility and hygroscopicity, which has significant value for future drug optimization and development.
Crystal Pharmaceutical (Suzhou) Co., Ltd.
C C A A A
C07B C07D A61P A61K A61K
additional inventional inventional inventional inventional
Fei Hui Xiaoyu Yuhao Minhua Yanfeng
Lu Gao Zhang Chen Chen Zhang