Dority & Manning, P.A.
4-substituted benzoxaborole compounds and uses thereof
Substituted benzoxaboroles whose structure comprises Formula (III), wherein R3 is selected from —CH3, —CH2CH3, —CH2═CH2, —CH2CH2CH3, —CH(CH3)2, —CH2CH2═CH2, and cyclopropyl, R1 and R2 are each independently selected from H, —CH3, —CH2CH3, —CH2CH2CH3, and —CH(CH3)2; compositions containing such compounds, their use in therapy, including their use as anti-mycobacterial agents, for example in the treatment of a mycobacterial infection in a mammal, and methods for the preparation of such compounds, are provided.
GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED ANACOR PHARMACEUTICALS, INC.
A A C A A A A A A A A A A A A C A A
A61P A61K C07B A61P A61P A61P A61P A61P A61P A61K A61P A61P A61P A61P A61P C07F A61P A61P
inventional inventional additional inventional inventional inventional inventional inventional inventional inventional inventional inventional inventional inventional inventional inventional inventional inventional
Carlos Michael Richard Kevin (Dickon) Vincent Jacob J. David Ilaria Xianfeng
Alemparte-Gallardo Alley Hernandez Plattner Barros-Aguirre Giordano Li